ECHC 2021

XXIX European Colloquium on Heterocyclic Chemistry

 Virtual Event    April 26-28, 2021

Keynote Lectures

Constructing Small Rings by Palladium(0)-catalyzed C-H Activation (KL03)

Prof. Olivier BAUDOIN
Prof. Olivier BAUDOIN
UNIVERSITY OF BASEL, Basel, Switzerland
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New Tools for the Introduction of Emergent Fluorinated Moieties (KL08)

Dr Tatiana BESSET
Dr Tatiana BESSET
INSA OF ROUEN, Mont-Saint-Aignan, France
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Three-Dimensional Heterocycles: Syntheses and Opportunities (KL01)

Prof. Carsten BOLM
Prof. Carsten BOLM
RWTH AACHEN, Aachen, Germany
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The Prebiotic Origin of the RNA Nucleosides (KL06)

Prof. Thomas CARELL
Prof. Thomas CARELL
LUDWIG-MAXIMILIANS-UNIVERSITY, München, Germany
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Alpha-Heterosubstituted Organolithiums: Swinging Between Carbanions and Carbenoids (KL13)

Prof. Saverio FLORIO
Prof. Saverio FLORIO
UNIVERSITY OF BARI "ALDO MORO", Bari, Italy
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Synthetic Biological and Synthetic Chemical Tools (Genochemetics) for Late Stage C-H Activation and Small Molecule Vectorisation (KL12)

Prof. Rebecca GOSS
Prof. Rebecca GOSS
UNIVERSITY OF ST ANDREWS, St Andrews, United Kingdom
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Cyclophanes, Cryptands and Supramolecular Polymers with Pyridine, Phenothiazine and Triazine Units (KL02)

Prof. Ion GROSU
Prof. Ion GROSU
BABES-BOLYAI UNIVERSITY, Cluj-Napoca, Romania
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Lewis Acid Enabled Novel Reactivities in Asymmetric Catalysis (KL05)

Prof. Syuzanna HARUTYUNYAN
Prof. Syuzanna HARUTYUNYAN
UNIVERSITY OF GRONINGEN, Groningen, The Netherlands
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Why do heterocycles make nice cores in drug discovery – the lesson of Mcl-1 inhibitors (KL11)

Dr Andras KOTSCHY
Dr Andras KOTSCHY
SERVIER RESEARCH INSTITUTE OF MEDICINAL CHEMISTRY, Budapest, Hungary
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Designing New Synthetic Concepts for Imparting Molecular Complexity with C-1 Sources (KL04)

Prof. Vittorio PACE
Prof. Vittorio PACE
UNIVERSITY OF TURIN, Turin, Italy
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Nickel Catalysis for C-C and C-heteroatom Bond Forming Reactions (KL10)

Prof. Magnus RUEPING
Prof. Magnus RUEPING
RWTH AACHEN, Aachen, Germany
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Springer Heterocyclic Chemistry Award Lecture
Some Adventures in Strategy-Guided Synthesis of Complex, Bioactive Natural Products (KL09)

Prof. Christopher VANDERWAL
Prof. Christopher VANDERWAL
UNIVERSITY OF CALIFORNIA, Irvine, United States
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Catalytic Asymmetric Cycloaddition to Access Chiral Heterocycles by Novel P-Ligands: From N-heterocycles to Silicon-stereogenic Silacycles (KL07)

Prof. Li-Wen XU
Prof. Li-Wen XU
HANGZHOU NORMAL UNIVERSITY, Hangzhou, China
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Invited Lectures

Diels-Alder cascades for the synthesis of fused N-heterocycles (IL01)

Dr Nicolas BLANCHARD
Dr Nicolas BLANCHARD
UNIVERSITY OF UPPER-ALSACE/CNRS, Mulhouse, France
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Supramolecular Multidentate Strategy Towards Enantioselective Anion-binding Catalysis (IL04)

Prof. Olga GARCIA MANCHENO
Prof. Olga GARCIA MANCHENO
UNIVERSITY OF MÜNSTER, Münster, Germany
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Blessed by N-Heterocyclic Carbenes: Olefin Metathesis Catalysis Story (IL08)

Prof. Karol GRELA
Prof. Karol GRELA
UNIVERSITY OF WARSAW, WARSAW, Poland
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Electro-Induced Isocyanide-Based Multicomponent Reactions (IL05)

Dr Laurence GRIMAUD
Dr Laurence GRIMAUD
ECOLE NORMALE SUPÉRIEURE, Paris, France
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Novel Reactivity in Hypervalent Iodine-Mediated Vinylations (IL06)

Prof. Berit OLOFSSON
Prof. Berit OLOFSSON
STOCKHOLM UNIVERSITY, Stockholm, Sweden
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C-S Bond Formation of N-fused Heterocycles via Metal and Photoredox Catalysis (IL03)

Dr Sandrine PIGUEL
Dr Sandrine PIGUEL
UNIVERSITY PARIS-SACLAY, Paris, France
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Exploring Palladium Catalysis in Deep Eutectic Solvents (IL09)

Prof. Antonio SALOMONE
Prof. Antonio SALOMONE
UNIVERSITY OF BARI "ALDO MORO", Bari, Italy
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Counterion Mediated Approaches to Controlling Axial Chirality (IL02)

Prof. Martin SMITH
Prof. Martin SMITH
UNIVERSITY OF OXFORD, Oxford, United Kingdom
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Dearomatization of Indoles for the Total Synthesis of Natural Products (IL07)

Dr Guillaume VINCENT
Dr Guillaume VINCENT
UNIVERSITY PARIS-SACLAY, Orsay, France
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Oral Communications - Session 1

Diastereoselective Synthesis of Nonplanar 3-Amino-1,2,4-Oxadiazine Heterocycle: Structure Revision of Alchornedine (OC04)

Dr Frédéric BIHEL
Dr Frédéric BIHEL
CNRS / UNIVERSITY OF STRASBOURG, Illkirch, France
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Development in Phosphiranium Ions Chemistry (OC09)

Mr Mohammad AHMAD
Mr Mohammad AHMAD
URCOM - UNIVERSITÉ DU HAVRE, Le Havre, France
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Straightforward Synthesis of Highly Substituted 6H-Benzo[C]Chromenes via a Diels-Alder/Aromatization Approach (OC16)

Mr Marco BALLAROTTO
Mr Marco BALLAROTTO
UNIVERSITÀ DEGLI STUDI DI PERUGIA, Perugia, Italy
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Novel Methodologies Towards the Synthesis of Saturated Heterocycles: The Silyl-Prins Cyclization (OC02)

Prof. Asuncion BARBERO
Prof. Asuncion BARBERO
UNIVERSITY OF VALLADOLID, Valladolid, Spain

Competitive Dearomatization of Benzene vs Pyridine: 1,3-Cycloaddition Followed by Suzuki-Miyaura Coupling on the Remaining Sulfonyloxyimine Functionality (OC05)

Mr Sami BEN SALAH
Mr Sami BEN SALAH
URCOM (UNIVESITY LE HAVRE NORMANDIE), Orléans, France
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Expanding the Chemical Diversity of Azaaurones: From Synthesis to Modulation of E/Z Isomerization (OC15)

Mr André CAMPANICO
Mr André CAMPANICO
I.MED.ULISBOA - FFULISBOA, Lisboa, Portugal
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Stereoselective Preparation of Saturated 2-Aryl Nitrogen-Containing Heterocycles (OC17)

Prof. Iain COLDHAM
Prof. Iain COLDHAM
UNIVERSITY OF SHEFFIELD, Sheffield, United Kingdom
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2- and 6-Purinylmagnesium Halides in Dichloromethane: Scope and Insights into the Solvent Influence on Anion Stability (OC10)

Dr Silvia GAZZOLA
Dr Silvia GAZZOLA
UNIVERSITY OF INSUBRIA, Como, Italy
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Synthesis of Five- and Six-Membered Heterocyclic Structures Based on Alkyl 3-Bromo-3-Nitroacrylates (OC13)

Mr Kirill GOMONOV
Mr Kirill GOMONOV
HERZEN STATE PEDAGOGICAL UNIVERSITY OF RUSSIA, Saint-Petersburg, Russia
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Synthesis of Organic Fluorophores Derived From Tetrazapentalene Scaffold : Study of their Spectroscopic Properties for a Potential Application In Energy Conversion (0C08)

Mr Vincent GUTIERREZ
Mr Vincent GUTIERREZ
UNIVERSITY OF ORLÉANS - ICOA, Orléans, France
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New Methods for the Synthesis of Subtituted 2-Pyridones (OC19)

Dr Zahira KIBOU
Dr Zahira KIBOU
LABORATOIRE DE CATALYSE ET SYNTHÈSE EN CHIMIE ORGANIQUE, , Tlemcen, Algerie
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Complementary Methods to Access Tetrahydrofurans and Tetrahydropyrans from Cyclopropanes: Fluorosulfoxoniums vs Trifilic Acid as Promoters (OC11)

Mr Augustin MANEL
Mr Augustin MANEL
CNRS - UNIVERSITÉ DE STRASBOURG, Strasbourg, France
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Rapid Assembly of Molecular Complexity from Simple Enamide Building Blocks (OC03)

Prof. Georg MANOLIKAKES
Prof. Georg MANOLIKAKES
TU KAISERSLAUTERN, Kaiserslautern, Germany
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Coherent Synchronization of The Oxidation Reactions of Pyridine Bases by “Green Oxidizing Agents” – H2O2 and N2O (OC01)

Prof. T. NAGIEV
Prof. T. NAGIEV
RESEARCH CENTER OF AZERBAIJAN NATIONAL ENCYCLOPEDIA, Baku, Azerbaijan

N-N Bond Formation with Heteroaromatic Amines: Mild Access to Tricycles [6-5-6] Derivatives (OC14)

Mr Moussa NDIAYE
Mr Moussa NDIAYE
ICOA, Orleans, France
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Synthesis of Highly Functionnalized Propellanes from Bicyclic Hydroxylactones (OC20)

Prof. Olivier PIVA
Prof. Olivier PIVA
UNIVERSITE LYON 1, VILLEURBANNE, France
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Expeditious and Practical Synthesis of Tertiary Alcohols from Esters Enabled by Highly Polarized Organometallic Compounds Under Aerobic Conditions in Deep Eutectic Solvents or Bulk Water (OC07)

Mr Andrea Francesca QUIVELLI
Mr Andrea Francesca QUIVELLI
UNIVERSITY OF BARI, Bari, Italy
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Synthesis of New Heteroaromatic Fluoroalkylcompounds via Deprotonation of -CHF2 (OC12)

Ms Laura SANTOS
Ms Laura SANTOS
UNIVERSITY OF STRASBOURG, Strasbourg, France
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Synthesis of Novel Classes Of 4’-Spirocycloalkyl Nucleoside Analogues (OC06)

Dr Guido VERNIEST
Dr Guido VERNIEST
JANSSEN PHARMACEUTICA, Beerse, Belgium
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Oral Communications - Session 2

Isocyanoacetates in the Synthesis of Heterocyclic Compounds (OC38)

Dr Sonia ABAS PRADES
Dr Sonia ABAS PRADES
UNIVERSITY OF LEEDS, Leeds, United Kingdom
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N-Acyliminium Ions Chemistry: Iron Activation and Synthesis of Novel Heterocyclic Compounds via [2+2+2] Sequence (OC41)

Mr Sidi Mohamed ABDALLAHI
Mr Sidi Mohamed ABDALLAHI
UNIVERSITÉ DU HAVRE, Le havre, France
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Conception of Enantioselectivite Domino Processes for the Synthesis of Highly Tunable N-Heterocyclic Compounds (OC39)

Mr ISMAIL ALAHYEN
Mr ISMAIL ALAHYEN
UNIVERSITY OF LE HAVRE, le Havre, France
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Construction of N-Fluoroalkyl Nitrogen Heterocycles from Fluoroalkyl Azides (OC34)

Dr Petr BEIER
Dr Petr BEIER
ACADEMY OF SCIENCES OF THE CZECH REPUBLIC, Prague, Czech Republic
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Hydrogen Isotope Exchange - The Simplest Late Stage Functionalization (OC33)

Dr Volker DERDAU
Dr Volker DERDAU
SANOFI GERMANY, Frankfurt, Germany
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Iridium-Catalyzed β-C(SP2) -H Borylation of Enamides-Efficient Access to GEM-Dihalogeno N-Heterocycles (OC40)

Mr Ismael DONDASSE
Mr Ismael DONDASSE
ICOA, Orléans, France
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Synthesis and Functionalizations of (Het)Arenes with Visible Light (OC43)

Dr Indrajit GHOSH
Dr Indrajit GHOSH
UNIVERSITY OF REGENSBURG, Regensburg, Germany
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Cobalt-Catalyzed Atropoenantioselective C-H Arylation of Indoles (OC42)

Mr Nicolas JACOB
Mr Nicolas JACOB
UNIVERSITY OF STRASBOURG, Strasbourg, France
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Meldrum’s Acid as a Useful Platform for Organocatalyzed Synthesis of Chiral Heterocyclic Fragments (OC46)

Mr Arthur LEBRÊNE
Mr Arthur LEBRÊNE
LABORATORY COBRA, Rouen, France
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Access to α/β-Dipeptides through the Diastereoselective Multicomponent Organocatalytic Synthesis of Isoxazolidin-5-Ones (OC49)

Dr Thomas MARTZEL
Dr Thomas MARTZEL
COBRA, Rouen, France
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One-Pot Cross Coupling/CH Functionalisation Reactions: Quinoline as a Substrate and Ligand through N-Pd Interaction and an Example of Reversible Oxidative Addition? (OC45)

Dr Gerard MCGLACKEN
Dr Gerard MCGLACKEN
UNIVERSITY COLLEGE CORK, Cork, Ireland
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Powerful Stereoselective Strategies to Nitrogen-Containing Heterocycles in One-Pot: Maximizing the Sequential Steps While Reducing the Operations (OC35)

Dr Sara MENINNO
Dr Sara MENINNO
UNIVERSITY OF SALERNO, Fisciano, Italy
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Chiral Ammonium Aryloxides as Nucleophilic Organocatalysts: Application to the Enantioselective Decarboxylative Protonation of Meldrum’s Acid Derivatives (OC47)

Dr Sylvain OUDEYER
Dr Sylvain OUDEYER
UNIVERSITY OF ROUEN, COBRA-IRCOF, Rouen, France
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Phytoremediation by Plants and Valorization of Phytofixed Metals as Heterogeneous Ecocatalyst's in the Synthesis Of Azaheterocyclic Scaffolds (OC44)

Ms Christine SAFI
Ms Christine SAFI
UNIVERSITY LE HAVRE, Le Havre, France
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CU-Catalyzed Oxidative Allylic C-H Arylation of Inexpensive Alkenes with (Hetero)Aryl Boronic Acids (OC51)

Prof. Cédric SCHNEIDER
Prof. Cédric SCHNEIDER
UNIVERSITY OF ROUEN, COBRA-IRCOF, Rouen, France
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C-H Functionalizations via Transient σ-Alkyl/Vinyl-Palladium (II) Intermediates Capture in Batch and Continuous-Flow (OC37)

Dr Upendra K. SHARMA
Dr Upendra K. SHARMA
UNIVERSITY OF LEUVEN (KU LEUVEN), Heverlee, Belgium
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New Applications of Proline to Organic Synthesis (OC32)

Prof. Dmitry TSVELIKHOVSKY
Prof. Dmitry TSVELIKHOVSKY
THE HEBREW UNIVERSITY OF JERUSALEM, Jerusalem, Israel

Total Syntheses of Aspidosperma Alkaloids Through Sequences of Cascade Reactions (OC50)

Dr Szilárd VARGA
Dr Szilárd VARGA
RESEARCH CENTRE FOR NATURAL SCIENCES, Budapest, Hungary
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Asymmetric Organocatalysis and Cascade Reactions in the Stereoselective Synthesis of Heterocyclic Scaffolds (OC36)

Dr Fabrizio VETICA
Dr Fabrizio VETICA
SAPIENZA UNIVERSITY OF ROME, Roma, Italy
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Photocatalytic Generation of Carbanions from Carbonyls & Thiolate Anions as Phtotocatalysts for Borylation of Substituted Arenes (OC48)

Mr Shun WANG
Mr Shun WANG
UNIVERSITY OF REGENSBURG, Regensburg, Germany
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Transition-Metal Catalyzed Carbonylative Synthesis of Heterocycles (OC31)

Dr Xiao-feng WU
Dr Xiao-feng WU
LEIBNIZ-INSTITUT FÜR KATALYSE E. V, Rostock, Germany

Oral Communications - Session 3

The Pyrimidine Ring: A Wonderful Platform for the Conception of Advanced Luminescent Materials (OC81)

Dr Sylvain ACHELLE
Dr Sylvain ACHELLE
UNIVERSITÉ DE RENNES 1, Pommerit jaudy, France
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Design and Scale-Up of Amphiphilic Cationic Meso-Imidazolyl Porphyrin-Based Photosensitizers for Development of Potential Antimicrobial Agents (OC69)

Ms Zoe ARNAUT
Ms Zoe ARNAUT
UNIVERSITY OF COIMBRA, Coimbra, Portugal
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Computational Design and Synthesis of Benzimidazole Derivatives for Potential E. Coli DNA Gyrase B Inhibition (OC63)

Mr Rafael AROSO
Mr Rafael AROSO
UNIVERSIDADE DE COIMBRA, Coimbra, Portugal
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2-(Diazobenzyl)Chromones: New Templates for Easy Pharmacophore Introduction (OC67)

Mr Vasco BATISTA
Mr Vasco BATISTA
UNIVERSITY OF AVEIRO, Aveiro, Portugal
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High-Efficient Synthesis of Imidazo[1,2-A]Pyrimidines (OC18)

Mrs Djamila BENZENINE
Mrs Djamila BENZENINE
AIN TÉMOUCHENT UNIVERSITY, Tlemcen, Algerie

UGI Reaction and Isatin: A “Fast-Track" for the Discovery of New Bioactive Oxindoles (OC64)

Mr Pedro BRANDAO
Mr Pedro BRANDAO
UNIVERSITY OF COIMBRA, Coimbra, Portugal
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Quenched Activity-Based Probes as New Chemical Tools to Analyse Serine Hydrolases (OC68)

Ms Rita FÉLIX
Ms Rita FÉLIX
IMED.ULISBOA - INSTITUTO DE INVESTIGAÇÃO DO MEDICAMENTO, Lisboa, Portugal
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Development of New Heterocyclic Necroptosis Inhibitors: Targeting RIPK1 (OC79)

Ms Lara FIDALGO
Ms Lara FIDALGO
FFULISBOA, Lisboa, Portugal
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APT Pro-Drug Inhibitors of Clostridiodes Difficile (OC77)

Dr William FRASER
Dr William FRASER
ASTON UNIVERSITY, Birmingham, United Kingdom
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Synthesis, Biological Evaluation and Binding Mode of New CLK1/DYRK1A Inhibitors Presenting a Pyrido[3,4-G]Quinazoline Moiety (OC61)

Dr Francis GIRAUD
Dr Francis GIRAUD
INSTITUTE OF CHEMISTRY OF CLERMONT-FERRAND, AUBIERE, France
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Microscope Laser Assisted Photooxidative Activation of Bioorthogonal Clickox Probes (OC80)

Ms Dora KERN
Ms Dora KERN
RESEARCH CENTRE FOR NATURAL SCIENCES, Budapest, Hungary
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Synthesis and Structure-Activity Relationship Studies of Antimalarial Thienopyrimidine Derivatives (OC72)

Mrs Prisca LAGARDÈRE
Mrs Prisca LAGARDÈRE
INSTITUT DES BIOMOLÉCULES MAX MOUSSERON, Montpellier, France
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Different Heterocycles, Distinct Affinities - Synthesis and Study of a Novel Class of Potent Necroptosis Inhibitors (OC76)

Mr André LUZ
Mr André LUZ
FACULTY OF PHARMACY, UNIVERSITY OF LISBON, Lagos, Portugal
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A Convenient Route to New (Radio)Fluorinated or (Radio)Iodinated TIC(OH) Analogues (OC78)

Dr Aurélie MAISONIAL BESSET
Dr Aurélie MAISONIAL BESSET
UMR 1240 IMOST - INSERM UNIVERSITE CLERMONT AUVERGNE, Clermont Ferrand, France
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1,3,4-Oxadiazole-Indole Hybrids: Synthesis and their Protective Activity Against Oxidative Stress (OC74)

Dr Vida MALINAUSKIENE
Dr Vida MALINAUSKIENE
KAUNAS UNIVERSITY OF TECHNOLOGY, Kaunas, Lithuania
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Synthesis and in-vitro Antiproliferative Studies of Pinane-Based Pyrimidine Derivatives (OC75)

Mr RAJI MOUNIR
Mr RAJI MOUNIR
UNIVERSITY OF SZEGED, Szeged, Hungary
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T-Shaped and Cruciform Donor-Acceptor Psoralen Fluorophores by Consecutive One-Pot Syntheses (OC65)

Prof. Thomas J. J. MÜLLER
Prof. Thomas J. J. MÜLLER
HEINRICH-HEINE-UNIVERSITÄT DÜSSELDORF, Düsseldorf, Germany
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Synthesis of Functionalized Tryptophan Derivatives and their Use in the Total Synthesis of Indole Alkaloid Natural Products (OC66)

Prof. GIOVANNI PIERSANTI
Prof. GIOVANNI PIERSANTI
UNIVERSITY OF URBINO, URBINO (PU), Italy
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Radiosynthesis Of [11C]EHT1610, A Potential Radioligand For Quantification Of Cerebral Dyrk1a By Pet Imaging (OC83)

Dr Pauline POUTREL
Dr Pauline POUTREL
CYCÉRON, Caen, France
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Hydroxylated Heterocycles as a Bioisosteric Tool to Modulate the Carboxylic Function into Design Potent Human Dihydroorotate Dehydrogenase Inhibitors (OC71)

Dr Stefano SAINAS
Dr Stefano SAINAS
UNIVERSITY OF TORINO, Torino, Italy
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Effect of Anchimeric Assistance in Chemistry of Phosphonium Enolates and its Application in Synthesis of a-Methylene-γ-Butyrolactone Derivatives with Cytotoxic Activity (OC62)

Prof. Alexey SALIN
Prof. Alexey SALIN
KAZAN FEDERAL UNIVERSITY, Kazan, Russia
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Design, Synthesis and Evaluation of Acridine Derivatives as Potential Leishmanial Inhibitors (OC70)

Mr Carlos SILVA
Mr Carlos SILVA
UNIVERSITY OF AVEIRO, Aveiro, Portugal
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Radiolabelled Porphyrin Metalla-Assemblies in Cellulose Nanocrystals, a Theranostic Agent for PDT (OC82)

Mr Joao SIMOES
Mr Joao SIMOES
BIOEMTECH, Athens, Greece

Ultrasound-Assisted One-Pot Green Synthesis of Novel Isoxazoline Derivatives of Thiazolidine-2,4-Dione and Antidiabetic Activity Investigation (OC73)

Ms Fatima Zahra THARI
Ms Fatima Zahra THARI
MOHAMMED V UNIVERSITY, Rabat, Morocco
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